Corticosteroid Class
Budesonide
Brand: Entocort EC (US/EU) / Budenofalk (EU) / Budecort (IN) / Budesonide (BD)
Subclass: High first-pass glucocorticoid
PK:
t½ 3 hours | Clearance: hepatic
Max Dose: 9 day
Max Dose: 9 day
moderate
AE: Adrenal suppression (less than prednisolone), edema, mood changes
AE: Adrenal suppression (less than prednisolone), edema, mood changes
Dexamethasone
Brand: Dexona
Subclass: Long-acting Glucocorticoid
PK:
t½ 48 hours | Clearance: hepatic
Max Dose: 16 day
Max Dose: 16 day
moderate
AE: Hyperglycemia, insomnia, muscle wasting
AE: Hyperglycemia, insomnia, muscle wasting
Hydrocortisone
Brand: Cortef
Subclass: Short-acting
PK:
t½ 1.5 hours | Clearance: hepatic
Max Dose: 240 day
Max Dose: 240 day
moderate
AE: Fluid retention, mood changes, adrenal suppression
AE: Fluid retention, mood changes, adrenal suppression
Prednisolone
Brand: Pred
Subclass: Glucocorticoid
PK:
t½ 3 hours | Clearance: hepatic
Max Dose: 60 day
Max Dose: 60 day
moderate
AE: Weight gain, mood changes, immunosuppression
AE: Weight gain, mood changes, immunosuppression