| Half-life | 40 days |
| Clearance Route | hepatic |
| Active Metabolites | no |
| Notes | IM monthly dosing; not daily mg concept; long half-life ~40 days. |
Severity: Moderate
Adverse Effects:
Injection site pain, liver enzyme elevation, hot flashes
Contraindications:
Severe hepatic impairment
Precautions:
Monitor LFTs; avoid pregnancy