| Half-life | 5 hours |
| Clearance Route | hepatic |
| Active Metabolites | none |
| Notes | Poorly absorbed (<15%); most drug stays in gut. Use with caution in hepatic impairment. |
Severity: Mild
Adverse Effects:
Nausea, abdominal cramps, diarrhea, dizziness, headache. Rare: elevated LFTs.
Contraindications:
Severe hepatic impairment
Precautions:
Avoid in pregnancy unless necessary; monitor LFTs if prolonged use; caution with piperazine (antagonistic).